Prof. Jean RODRIGUEZ
Prof.
Jean
RODRIGUEZ
AMU iSm2 Service 531
Campus Scientifique de St Jérôme
13397
Marseille cedex 20
Téléphone :
Fax :
0491 28 9187
Courriel :
Parcours :
1984 : PhD of Speciality at the University of Aix-Marseille
1984 : Recruted by the CNRS as Attaché de Recherche
1987 : PhD in Sciences at the University of Aix-Marseille
1988 : Postdoctoral reseach associate, University of California (Berkeley), supervisor: Prof K.P.C. Vollhardt
1989 : Promoted Chargé de Recherche de 1ère classe at CNRS
1992 : Habilitation at the University of Aix-Marseille
1998 : Promoted Directeur de Recherche at the CNRS
2002 : Nominated full Professor at the University of Aix-Marseille
Distinctions :
1998 : Prize from ACROS-French Chemical Society in organic chemistry 2009 : Prize from the Société Chimique de France, Division Chimie Organique 2013 : Member of the Editorial Board of European Journal of Organic Chemistry 2013 : Distinguished Senior Member of the Société Chimique de France 2013 : Dr Paul Janssen invited lecturer, Beerse (Belgium)
Enseignements :
Bachelor Degree in Chemistry
*Ionic and Polar Rearrangements in Organic Synthesis
Master Degree in Chemistry
*Strategies in Synthetic Organic Chemistry (Retrosynthetic analysis, Total synthesis, Protection and Deprotection of functional groups)
*New Selective Multiple Bond-Forming Transformations (Metallo- and Organocatalyzed Consecutive, Domino and Multicomponent reactions)
*Recent Applications of enantioselective metallo- and organocatalysis in Organic Synthesis
Collaborations et groupes :
Dr Damien BONNE, Assistant Professor
Dr Xavier BUGAUT, Assistant Professor
Dr Thierry CONSTANTIEUX, Full Professor
Dr Yoann COQUEREL, Associate Researcher from the CNRS
Dr Adrien QUINTARD, Associate Researcher from the CNRS
Dr Rodolphe BEAU, Postdoctoral Reseach Associate (2016-2018)
Dr Nicolas DALMASSO, Postdoctoral Associate (2016-2018)
Yasmin REVIVOT, PhD student (2017-2020)
Peng LIU, PhD student (2017-2020)
Brian CASTRO, PhD student (2017-2020)
Céline SPERANDIO, PhD student (2016-2019)
Yun-Long WEI PhD student (2015-2018)
Responsabilités administratives :
1999-2007 : Member of Bureau National de la S F C, Division Chimie Organique
2000-2006 : Expert auprès du ministère dans le cadre de la MSTP4
2004-2007 : Director of the Reseach Unit SYMBIO
2006-2011 : Chargé de Mission à l'Institut de chimie du CNRS (section 12)
2008- Present : Director of the Institut des Sciences Moléculaires de Marseille (iSm2)
Publications (210)
Reference
Résumé graphique
HAL
Synthetic Studies on the MARDi Cascade: Stereoselective Synthesis of Heterocyclic Seven-Membered Rings
Yoann Coquerel, David Bensa, Alain Doutheau, Jean Rodriguez, Organic Letters, 2006, 8, 4819-4822. <hal-02989798>
✖
An Operationally Simple Base-Catalyzed Multi- component Domino Transfor-mation: Stereoselective Preparation of Trisubstituted Alkenes and 1,3-Dienes.
Hadjira Habib-Zahmani, Salih Hacini, Cédric Bories, Robert Faure, Jean Rodriguez Synthesis 2005, 2151-2156
✖
Azaindoles: Provence Technologies et PCAS sallient.
Jean Rodriguez Industrie Pharma Magazine2005, 17, 10.
✖
Aliphatic and Alicyclic Ketones (except Cyclobutanones and Cyclopropanones): Synthesis by Fragmentation and Rearrangement
T. Constantieux, J. Rodriguez. Science of Synthesis, Volume 26, J. Cossy, Ed., Georg Thieme Verlag (Stuttgart), 2005, 413-462.
✖
Unique Michael Addition-Initiated Domino Reaction for the Stereoselective Synthesis of Functionalized Macrolactones from r-Nitroketones in Water
Giorgio Giorgi, Sonia Miranda, Pilar Lopez-Alvarado, Carmen Avendano, Jean Rodriguez and J. Carlos Menendez. Org. Lett. 2005, 7, 2197-2200
✖
Azaindoles: Provence Technologies et PCAS mettent leurs forces en commun.
Jean Rodriguez Chimie Pharma Hebdo2005, 312, 4.
✖
Multicomponent Reactions with 1,3-Dicarbonyl Derivatives: Applications to the Synthesis of Polyfunctionalized Heterocycles.
T. Constantieux, J. Rodriguez dans : « Targets in Heterocyclic Systems » Vol 9, 2005.
✖
Azaindoles as medicinally relevant scaffolds.
J. Rodriguez, M. Feraud Spec. Chem. Mag.2005, 12, 16.
✖
Multicomponent Domino Reaction from b-Ketoamides: Highly Efficient Access to Original Polyfunctionalized 2,6-Diazabicyclo[2.2.2]octane Cores.
Frédéric Liéby-Muller, Thierry Constantieux, and Jean Rodriguez J. Am. Chem. Soc. 2005, 127, 17176-17177.
✖
P-BEMP: a New Efficient and Commercially Available User-friendly and Recyclable Heterogeneous Organocatalyst for the Michael Addition of 1,3-Dicarbonyl Compounds.
D. Bensa, T. Constantieux, J. Rodriguez. Synthesis, 2004, 923-027
✖
Pages
Ouvrages (3)
Reference
Résumé graphique
HAL
Stereoselective Multiple Bond-Forming Transformations in Organic Synthesis
Eds.: J. Rodriguez, D. Bonne, John Wiley & Sons, Inc., Hoboken, NJ, USA, 2015.
✖
Jean Rodriguez, Damien Bonne. Stereoselective Multiple Bond-Forming Transformations in Organic Synthesis. John Wiley & Sons, 2015, 978-1-118-67271-6. ⟨hal-01323433⟩
✖
1-Nitrocyclohexene
David Pierrot, Damien Bonne, Jean Rodriguez 2014, e-EROS Encyclopedia of Reagents for Organic Synthesis. 15.
✖
Chapitres d'ouvrages (9)
Reference
Résumé graphique
HAL
Yoann Coquerel, Jean Rodriguez. The Wolff Rearrangement: Tactics, Strategies and Recent Applications in Organic Synthesis. Molecular Rearrangements in Organic Synthesis, Johne Wiley & Sons, pp.59-84, 2015, 978-1-118-34796-6. ⟨hal-01224316⟩
✖
1,3-Dicarbonyls in Multicomponent Reactions
X. Bugaut, T. Constantieux, Y. Coquerel, J. Rodriguez, In Multicomponent Reactions in Organic Synthesis, Eds.: J. Zhu, Q. Wang, M.-X. Wang, Wiley-VCH, Weinheim, 2014, Chap. 5, pp 109-158.
✖
Xavier Bugaut, Thierry Constantieux, Yoann Coquerel, Jean Rodriguez. 1,3-Dicarbonyls in Multicomponent Reactions. J. Zhu, Q. Wang, M.-X. Wang. Multicomponent Reactions in Organic Synthesis, Wiley-VCH, Weinheim, pp.109-158, 2014, 978-3-527-33237-3. ⟨hal-01133604⟩
✖
Reactions Involving an alpha,beta-Unsaturated Compound as Electrophilic Component with the Michael Addition as the Key Step
J. Rodriguez, D. Bonne, Y. Coquerel, T. Constantieux, dans 'Multicomponent Reactions 2', 'Science of Synthesis Reference Library', T. J. J. Müller, Ed., Thieme, Stuttgart, 2013, Chap. 2.1.1, p. 1-36.
✖
Stereoselective Multicomponent Reactions: from Simple 1,3-Dicarbonyls to Functionalized Chiral Heterocycles
D. Bonne, Y. Coquerel, T. Constantieux, J. Rodriguez in Targets in Heterocyclic Systems - Chemistry and Properties, Vol. 15, Eds.: O. A. Attanasi, D. Spinelli, Societa? Chimica Italiana, Roma, 2011, pp. 140-163.
✖
Utilisation des dérivés 1,3-dicarbonylés dans les réactions domino et multicomposé
Damien Bonne, Thierry Constantieux, Yoann Coquerel, Jean Rodriguez Techniques de l'Ingénieur 2010, CHV2210
✖
Damien Bonne, Thierry Constantieux, Yoann Coquerel, Jean Rodriguez. Utilisation des dérivés 1,3-dicarbonylés dans les réactions domino et multicomposé. Ideas in Chemistry and Molecular Sciences: Advances in Synthetic Chemistry, pp.CHV2210, 2010. ⟨hal-00680619⟩
✖
Yoann Coquerel, Thomas Boddaert, Marc Presset, Damien Mailhol, Jean Rodriguez. Multiple Bond-Forming Transformations: the Key Concept towards Eco-compatible Synthetic Organic Chemistry. Ideas in Chemistry and Molecular Sciences, Vol.1 Advances in synthetic chemistry, Wiley-VCH, Weinheim, pp.187-202, 2010, 3527325395. ⟨hal-00681017⟩
✖
Maria del Mar Sanchez Duque, Christophe Allais, Nicolas Isambert, Thierry Constantieux, Jean Rodriguez. beta-diketo building blocks for MCRs-based syntheses of heterocycles. Topics in Heterocyclic Chemistry, Springer, pp.227-277, 2010, ⟨10.1007/7081_2010_26⟩. ⟨hal-00680508⟩
✓
Brevets (1)
Reference
Résumé graphique
HAL
Adrien Quintard, Céline Sperandio, Jean Rodriguez. NOVEL FLUORINATED POLYOLS AND THEIR USE AS ORGANOGELATORS. France, Patent n° : WO/2019/238582. 2019. ⟨hal-02878986⟩
✖
Prof.
Jean
RODRIGUEZ
Prof.
Jean
RODRIGUEZ
AMU iSm2 Service 531
Campus Scientifique de St Jérôme
13397
Marseille cedex 20
Téléphone :
Fax :
0491 28 9187
Courriel :
Parcours :
1984 : PhD of Speciality at the University of Aix-Marseille
1984 : Recruted by the CNRS as Attaché de Recherche
1987 : PhD in Sciences at the University of Aix-Marseille
1988 : Postdoctoral reseach associate, University of California (Berkeley), supervisor: Prof K.P.C. Vollhardt
1989 : Promoted Chargé de Recherche de 1ère classe at CNRS
1992 : Habilitation at the University of Aix-Marseille
1998 : Promoted Directeur de Recherche at the CNRS
2002 : Nominated full Professor at the University of Aix-Marseille
Distinctions :
1998 : Prize from ACROS-French Chemical Society in organic chemistry 2009 : Prize from the Société Chimique de France, Division Chimie Organique 2013 : Member of the Editorial Board of European Journal of Organic Chemistry 2013 : Distinguished Senior Member of the Société Chimique de France 2013 : Dr Paul Janssen invited lecturer, Beerse (Belgium)
Enseignements :
Bachelor Degree in Chemistry
*Ionic and Polar Rearrangements in Organic Synthesis
Master Degree in Chemistry
*Strategies in Synthetic Organic Chemistry (Retrosynthetic analysis, Total synthesis, Protection and Deprotection of functional groups)
*New Selective Multiple Bond-Forming Transformations (Metallo- and Organocatalyzed Consecutive, Domino and Multicomponent reactions)
*Recent Applications of enantioselective metallo- and organocatalysis in Organic Synthesis
Collaborations et groupes :
Dr Damien BONNE, Assistant Professor
Dr Xavier BUGAUT, Assistant Professor
Dr Thierry CONSTANTIEUX, Full Professor
Dr Yoann COQUEREL, Associate Researcher from the CNRS
Dr Adrien QUINTARD, Associate Researcher from the CNRS
Dr Rodolphe BEAU, Postdoctoral Reseach Associate (2016-2018)
Dr Nicolas DALMASSO, Postdoctoral Associate (2016-2018)
Yasmin REVIVOT, PhD student (2017-2020)
Peng LIU, PhD student (2017-2020)
Brian CASTRO, PhD student (2017-2020)
Céline SPERANDIO, PhD student (2016-2019)
Yun-Long WEI PhD student (2015-2018)
Responsabilités administratives :
1999-2007 : Member of Bureau National de la S F C, Division Chimie Organique
2000-2006 : Expert auprès du ministère dans le cadre de la MSTP4
2004-2007 : Director of the Reseach Unit SYMBIO
2006-2011 : Chargé de Mission à l'Institut de chimie du CNRS (section 12)
2008- Present : Director of the Institut des Sciences Moléculaires de Marseille (iSm2)
Publications (210)
| Reference | Résumé graphique | HAL |
|---|---|---|
|
Synthetic Studies on the MARDi Cascade: Stereoselective Synthesis of Heterocyclic Seven-Membered Rings |
|
✖ |
|
An Operationally Simple Base-Catalyzed Multi- component Domino Transfor-mation: Stereoselective Preparation of Trisubstituted Alkenes and 1,3-Dienes. |
|
✖ |
|
Azaindoles: Provence Technologies et PCAS sallient. |
|
✖ |
|
Aliphatic and Alicyclic Ketones (except Cyclobutanones and Cyclopropanones): Synthesis by Fragmentation and Rearrangement |
|
✖ |
|
Unique Michael Addition-Initiated Domino Reaction for the Stereoselective Synthesis of Functionalized Macrolactones from r-Nitroketones in Water |
|
✖ |
|
Azaindoles: Provence Technologies et PCAS mettent leurs forces en commun. |
|
✖ |
|
Multicomponent Reactions with 1,3-Dicarbonyl Derivatives: Applications to the Synthesis of Polyfunctionalized Heterocycles. |
|
✖ |
|
Azaindoles as medicinally relevant scaffolds. |
|
✖ |
|
Multicomponent Domino Reaction from b-Ketoamides: Highly Efficient Access to Original Polyfunctionalized 2,6-Diazabicyclo[2.2.2]octane Cores. |
|
✖ |
|
P-BEMP: a New Efficient and Commercially Available User-friendly and Recyclable Heterogeneous Organocatalyst for the Michael Addition of 1,3-Dicarbonyl Compounds. |
|
✖ |
Pages
Ouvrages (3)
| Reference | Résumé graphique | HAL |
|---|---|---|
|
Stereoselective Multiple Bond-Forming Transformations in Organic Synthesis |
|
✖ |
|
Jean Rodriguez, Damien Bonne. Stereoselective Multiple Bond-Forming Transformations in Organic Synthesis. John Wiley & Sons, 2015, 978-1-118-67271-6. ⟨hal-01323433⟩ |
|
✖ |
|
1-Nitrocyclohexene |
|
✖ |
Chapitres d'ouvrages (9)
| Reference | Résumé graphique | HAL |
|---|---|---|
|
Yoann Coquerel, Jean Rodriguez. The Wolff Rearrangement: Tactics, Strategies and Recent Applications in Organic Synthesis. Molecular Rearrangements in Organic Synthesis, Johne Wiley & Sons, pp.59-84, 2015, 978-1-118-34796-6. ⟨hal-01224316⟩ |
|
✖ |
|
1,3-Dicarbonyls in Multicomponent Reactions |
|
✖ |
|
Xavier Bugaut, Thierry Constantieux, Yoann Coquerel, Jean Rodriguez. 1,3-Dicarbonyls in Multicomponent Reactions. J. Zhu, Q. Wang, M.-X. Wang. Multicomponent Reactions in Organic Synthesis, Wiley-VCH, Weinheim, pp.109-158, 2014, 978-3-527-33237-3. ⟨hal-01133604⟩ |
|
✖ |
|
Reactions Involving an alpha,beta-Unsaturated Compound as Electrophilic Component with the Michael Addition as the Key Step |
|
✖ |
|
Stereoselective Multicomponent Reactions: from Simple 1,3-Dicarbonyls to Functionalized Chiral Heterocycles |
|
✖ |
|
Utilisation des dérivés 1,3-dicarbonylés dans les réactions domino et multicomposé |
|
✖ |
|
Damien Bonne, Thierry Constantieux, Yoann Coquerel, Jean Rodriguez. Utilisation des dérivés 1,3-dicarbonylés dans les réactions domino et multicomposé. Ideas in Chemistry and Molecular Sciences: Advances in Synthetic Chemistry, pp.CHV2210, 2010. ⟨hal-00680619⟩ |
|
✖ |
|
Yoann Coquerel, Thomas Boddaert, Marc Presset, Damien Mailhol, Jean Rodriguez. Multiple Bond-Forming Transformations: the Key Concept towards Eco-compatible Synthetic Organic Chemistry. Ideas in Chemistry and Molecular Sciences, Vol.1 Advances in synthetic chemistry, Wiley-VCH, Weinheim, pp.187-202, 2010, 3527325395. ⟨hal-00681017⟩ |
|
✖ |
|
Maria del Mar Sanchez Duque, Christophe Allais, Nicolas Isambert, Thierry Constantieux, Jean Rodriguez. beta-diketo building blocks for MCRs-based syntheses of heterocycles. Topics in Heterocyclic Chemistry, Springer, pp.227-277, 2010, ⟨10.1007/7081_2010_26⟩. ⟨hal-00680508⟩ |
|
✓ |
Brevets (1)
| Reference | Résumé graphique | HAL |
|---|---|---|
|
Adrien Quintard, Céline Sperandio, Jean Rodriguez. NOVEL FLUORINATED POLYOLS AND THEIR USE AS ORGANOGELATORS. France, Patent n° : WO/2019/238582. 2019. ⟨hal-02878986⟩ |
|
✖ |