Institut des Sciences Moléculaires de Marseille Université Paul cézanne Aix Marseille III

               
       
Boite à outil Stéréo

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

 

les 172 publications de Stéréo

Some papers are available on the Hyper Articles on Line (HAL) here or on HAL-AMU

Title - Authors - Journal
Graphical Abstracts
Catalytic Enantioselective Desymmetrization of Meso Compounds in Total Synthesis of Natural Products: Towards an Economy of Chiral Reagents

J. Merad, M. Candy, J.-M. Pons, C. Bressy Synthesis 2017, accepted (invited review) DOI: 10.1055/s-0036-1589493

Tunable Copper-Catalyzed Multicomponent Reaction Towards Alkaloid-Inspired Indole/Lactam Polycycles

M. I. D. MARDJAN, S. PERIE, J.-L. PARRAIN and L. COMMEIRAS, Organic & Biomolecular Chemistry, 2017, DOI: 10.1039/C7OB00532F

L'éco-conception, un défi pour la recherche fondamentale

"A. Quintard, X. Bugaut, T. Constantieux, in "" Economie circulaire et territoires"". Eds: Y. Lazzeri, D. _Bonnet, M. Domeizel, Presses universitaires d'Aix-Marseille, 2017, p133-138. "

Enantioselective Syntheses of Furan Atropisomers by an Oxidative Central-to-Axial Chirality Conversion Strategy

Vivek S. Raut, Marion Jean, Nicolas Vanthuyne, Christian Roussel, Thierry Constantieux, Cyril Bressy, Xavier Bugaut, Damien Bonne, and Jean Rodriguez J. Am. Chem. Soc., 2017, 139 (6), 2140?2143

Enantioselective Organocatalyzed Consecutive Synthesis of Alkyl 4,5-Dihydrofuran-2-carboxylates from alpha-Keto Esters and (Z)-beta-Chloro-?-nitrostyrenes

Diana Becerra, Wilfried Raimondi, Daniel Dauzonne, Thierry Constantieux, Damien Bonne, Jean Rodriguez Synthesis 2017, 49(01), 195-201

Organocatalytic Multicomponent Reactions of 1,3-Dicarbonyls for the Synthesis of Enantioenriched Heterocycles

H. Du, Y. Dudognon, M. M. Sanchez Duque, S. Goudedranche, D. Bonne, J. Rodriguez, X. Bugaut, T. Constantieux Synthesis, 2016, 48, 3479-3503.

From Simple Cyclic 1,3-Ketoamides to Complex Spirolactams by Supported Heterogeneous Organocatalysis with PS-BEMP

A. Benmaati, H. Habib Zahmani, S. Hacini, J. C. Menéndez, X. Bugaut, J. Rodriguez, T. Constantieux Synthesis, 2016, 48, 3217-3231.

Polyketides

F. Schaefers, T. A. M. Gulder, C. Bressy, M. Smietana, E. Benedetti, S. Arseniyadis, M. Kalesse, and M. Cordes. Chap 2, pp 21-129 in From Biosynthesis to Total Synthesis: Strategies and Tactics for Natural Products, A. Zografos (Ed.), Wiley, 2016.

Catalytic Scanning Probe Nanolithography (cSPL): Control of the AFM Parameters in Order to Achieve Sub-100-nm Spatially Resolved Epoxidation of Alkenes Grafted onto a Surface

Mesquita, J. Botton, D. A. Valyaev, C. François, L. Patrone, T. S. Balaban, M. Abel, J.-L. Parrain, O. Chuzel, S. Clair, Langmuir 2016, 32, 4034-4042.

Straightforward and Controlled Shape Access to Efficient Macrocyclic Imidazolylboronium Anion Receptors

M. Toure, L. Charles, C. Chendo, S. Viel, O. Chuzel, J.-L. Parrain, Chem. Eur. J. 2016, 22, 8937?8942

Enantioselective Catalysis by Chiral Isothioureas

J. Merad, J.-M. Pons, O. Chuzel, C. Bressy, Eur. J. Org. Chem. 2016, 5589-5610.

A switchable dual organocatalytic system and the enantioselective total synthesis of the quadrane sesquiterpene suberosanone

Y. Ren, Marc Presset, Jeremy Godemert, Nicolas Vanthuyne, Jean-Valère Naubron, Michel Giorgi, Jean Rodriguez, and Yoann Coquerel Chem. Commun. 2016, 52, 6565-6568

Time-Efficient Synthesis of Pyrido[2,3-d]pyrimidinones via alpha-Oxoketenes

Juan-Carlos Castillo, Jairo Quiroga, Jean Rodriguez, and Yoann Coquerel Eur. J. Org. Chem. 2016, 1994-1999

Recent Achievements in Enantioselective Borrowing Hydrogen by the Combination of Iron- and Organocatalysis

Mylène Roudier, Thierry Constantieux, Jean Rodriguez, and Adrien Quintard Chimia 2016, 70, 97?101

Copper(I)-Catalysed Multicomponent Reaction: Straightforward Access to 5-Hydroxy-1H-pyrrol-2(5H)-ones

Muhammad Idham Darussalam Mardjan, Jean-Luc Parrain andLaurent Commeiras Adv. Synth. Catal. 2016 DOI: 10.1002/adsc.201500994

Addition of Silylated Nucleophiles to ?-Oxoketenes

Y. Dudognon, M. Presset, J. Rodriguez, Y. Coquerel, X. Bugaut, T. Constantieux Chem. Commun. 2016, 52, 3010-3013.

Combining Organocatalysis with Central-to-Axial Chirality Conversion: Atroposelective Hantzsch-Type Synthesis of 4-Arylpyridines

O. Quinonero, M. Jean, N. Vanthuyne, C. Roussel, D. Bonne, T. Constantieux, C. Bressy, X. Bugaut, J. Rodriguez Angew. Chem. Int. Ed. 2016, 55,1401-1405.

Stereoselective Multiple Bond-Forming Transformations in Organic Synthesis

Eds.: J. Rodriguez, D. Bonne, John Wiley & Sons, Inc., Hoboken, NJ, USA, 2015.

Pseudo-Multicomponent Reactions of Arynes with N?Aryl Imines

Juan-Carlos Castillo, Jairo Quiroga, Rodrigo Abonia, Jean Rodriguez, Yoann Coquerel, J. Org. Chem. 2015, 80, 9767.

The Aryne aza-Diels?Alder Reaction: Flexible Syntheses of Isoquinolines

Juan-Carlos Castillo, Jairo Quiroga, Rodrigo Abonia, Jean Rodriguez, Yoann Coquerel, Org. Lett. 2015, 17, 3374-3377.

Enamine Activation of beta-Ketocarbonyls: New Opportunities in Enantioselective Organocatalysis

Jean Rodriguez and Yoann Coquerel ChemCatChem 2015, 7, 1263-1264.

Enantioselective Synthesis of Medium-Sized-Ring Lactones by Organocatalytic Michael Addition Followed by Reductively Initiated Fragmentation

Mylène Roudier, Thierry Constantieux, Adrien Quintard, Jean Rodriguez, 2015, Eur. J. Org. Chem. 2015, 5709,

Exploiting the Reactivity of 1,2-Ketoamides: Enantioselective Synthesis of Functionalized Pyrrolidines and Pyrrolo-1,4-benzodiazepine-2,5-diones

Paola Acosta, Diana Becerra, Sébastien Goudedranche, Jairo Quiroga, Thierry Constantieux, Damien Bonne, Jean Rodriguez Synlett 2015, 26, 1591?1595

Synergistic Cuamine catalysis for the enantioselective synthesis of chiral cyclohexenones

Adrien Quintard and Jean Rodriguez, Chem. Commun. 2015, 51, 9523.

Highly Enantioselective Acylation of Acyclic Meso 1,3-Diols through Synergistic Isothiourea-Catalyzed Desymmetrization/Chiroablative Kinetic Resolution

Je?re?my Merad, Prashant Borkar, Tracy Bouyon Yenda, Christèle Roux, Jean-Marc Pons, Jean-Luc Parrain, Olivier Chuzel, and Cyril Bressy, Org. Lett. 2015, 17, 2118-2121

The Wolff Rearrangement: Tactics, Strategies and Recent Applications in Organic Synthesis

Y. Coquerel, J. Rodriguez, In Molecular Rearrangements in Organic Synthesis, Ed.: C. Rojas, John Wiley & Sons, Hoboken, NJ, 2015, Chap 3, pp. 59-84.

Origin of the Enantioselectivity in Organocatalytic Michael Additions of beta-Ketoamides to alpha,beta-Unsaturated Carbonyls: A Combined Experimental, Spectroscopic and Theoretical Study

A. Quintard, D. Cheshmedzhieva, M. M. Sanchez?Duque, A.Gaudel-Siri, J.-V. Naubron, Y. Génisson, J.-C. Plaquevent, X. Bugaut, J. Rodriguez, T. Constantieux, Chem. Eur. J. 2015, 21, 778.

A Stable N-Heterocyclic Carbene Organocatalyst for Hydrogen/Deuterium Exchange Reactions between Pseudo-acids and Deuterated Chloroform

F. Perez, Y. Ren, T. Boddaert, J. Rodriguez, Y. Coquerel, J. Org. Chem. 2015, 80, 1092-1097,.

Metal-Free Multicomponent Syntheses of Pyridines

C. Allais, J.-M. Grassot, J. Rodriguez, T. Constantieux, Chem. Rev. 2014, 114, 10829-10868.

1,3-Dicarbonyls in Multicomponent Reactions

X. Bugaut, T. Constantieux, Y. Coquerel, J. Rodriguez, In Multicomponent Reactions in Organic Synthesis, Eds.: J. Zhu, Q. Wang, M.-X. Wang, Wiley-VCH, Weinheim, 2014, Chap. 5, pp 109-158.

Divergent Chemo-­, Regio?, and Diastereoselective Normal Electron-Demand Povarov-Type Reactions with alpha-Oxo-ketene Dienophiles

J. Galvez, J.-C. Castillo, J. Quiroga, M. Rajzmann, J. Rodriguez, Y. Coquerel, Org. Lett. 2014, 16, 4126-4129.

N-Heterocyclic Carbene-Catalyzed Carba-, Sulfa- and Phospha-Michael Additions with NHC?CO2 Adducts as Precatalysts

M. Hans, L. Delaude, J. Rodriguez, Y. Coquerel, J. Org. Chem. 2014, 79, 2758-2764.

A temporary-bridge strategy for enantioselective organocatalyzed synthesis of aza-seven-membered rings

Sébastien Goudedranche, David Pierrot, Thierry Constantieux, Damien Bonne and Jean Rodriguez Chem. Commun., 2014, 50 (98), 15605 - 15608

1-Nitrocyclohexene

David Pierrot, Damien Bonne, Jean Rodriguez 2014, e-EROS Encyclopedia of Reagents for Organic Synthesis. 1?5.

Organocatalytic Enantioselective Construction of Polyaromatic Architectures

Ophélie Quinonero, Dr. Cyril Bressy andDr. Xavier Bugaut Angew. Chem. Int. Ed. 2014, 53, 10861-10863.

Iron Cyclopentadienone Complexes: Discovery, Properties, and Catalytic Reactivity

A. Quintard, J. Rodriguez Angew. Chem. Int. Ed. 2014, 53, 4044-4055.

trans-1,2-Disiloxybenzocyclobutene, an adequate partner for the auto-oxidation: EPR/spin trapping and theoretical studies

Drujon J., Rahmani R., Héran V., Blanc R., Carissan Y., Tuccio B., Commeiras L., Parrain J.-L. Phys. Chem. Chem. Phys. 2014, 16, 7513-7520

Preyssler Heteropoly Acids Encapsulated in a Silica Framework for an ­Efficient Preparation of Fluorinated Hexahydropyrimidine Derivatives under Solvent-Free Conditions

Ángel G. Sathicq, Diego M. Ruiz, Tierry Constantieux, Jean Rodriguez, Gustavo P. Romanelli Synlett 2014, 25(6), 881-883,

Benzoin and Aza-Benzoin

Xavier Bugaut, In: Gary A. Molander and Paul Knochel (eds.), Comprehensive Organic Synthesis, 2nd Edition, Vol 1, Oxford: Elsevier, 2014, pp.424-470.

Organocatalytic Enantioselective Multicomponent Synthesis of Pyrrolopiperazines

H. Du, J. Rodriguez, X. Bugaut, T. Constantieux Adv. Synth. Catal. 2014, 356, 851-856,

Stereocontrol of All-Carbon Quaternary Centers through Enantioselective Desymmetrization of Meso Primary Diols by Organocatalyzed Acyl Transfer

Christèle Roux, Mathieu Candy, Jean-Marc Pons, Olivier Chuzel, and Cyril Bressy, Angew. Chem. Int. Ed. 2014, 53, 766 -770

alpha,beta-Unsaturated Acyl Cyanides as New Bis-Electrophiles for Enantioselective Organocatalyzed Formal [3+3] Spiroannulation

S. Goudedranche, X. Bugaut, T. Constantieux, D. Bonne, J. Rodriguez, Chem. Eur. J. 2014, 20, 410-415. (Highlighted in Synform, 2014, 4, A49)

Macrocyclic compounds and their use for trapping anions

Parrain Jean-Luc, Chuzel Olivier, Toure Momar From PCT Int. Appl. (2014), WO 2014206931 A1 20141231

Enantioselective Organocatalytic Multicomponent Synthesis of 2,6-Diazabicyclo[2.2.2]octanones

M. M. Sanchez Duque, O. Baslé, Y. Génisson, J.-C. Plaquevent, X. Bugaut, T. Constantieux, J. Rodriguez, Angew. Chem. Int. Ed. 2013, 52, 14143-14146. (Highlighted in Synfacts, 2014, 10, 137),

Design, Synthesis, and Organocatalytic Activity of N-Heterocyclic Carbenes Functionalized with Hydrogen-Bond Donors in Enantioselective Reactions of Homoenolates

Faisal Nawaz, Mehdi Zaghouani, Damien Bonne, Olivier Chuzel, Jean Rodriguez, and Yoann Coquerel Eur. J. Org. Chem. 2013, 8253-8264.

Temporary Intramolecular Generation of Pyridine Carbenes in Metal-Free Three-Component C_H Bond Functionalisation/Aryl-Transfer Reactions

Faisal Nawaz, Kishor Mohanan, Laurence Charles, Michel Rajzmann, Damien Bonne, Olivier Chuzel, Jean Rodriguez, and Yoann Coquerel Chem. Eur. J. 2013, 19, 17578 - 17583.

An Iron/Amine-Catalyzed Cascade Process for the Enantioselective Functionalization of Allylic Alcohols

A. Quintard, T. Constantieux, J. Rodriguez, Angew. Chem. Int. Ed. 2013, 52, 12883-12887.

Book chapter: Organocatalytic Conjugate Addition in Stereoselective Synthesis

A. Quintard, A. Alexakis, in 'Stereoselective Synthesis of Drugs and Natural Products'. Eds: V. Andrushko, N. Andrushko, Wiley- Blackwell, Hoboken, NJ, 2013, Chap. 11.

Addition to Nitroolefins and Vinyl Sulfones

Christele Roux, Cyril Bressy, Chap. 34, pp 1013-1042 in Comprehensive Enantioselective Organocatalysis: Catalysts, Reactions, and Applications, Vol. 3, P. I. Dalko (Ed.), Wiley VCH, Weinheim, 2013

Grafting a homogeneous transition metal catalyst onto a silicon AFM probe: a promising strategy for chemically constructive nanolithography

Dmitry A. Valyaev, Sylvain Clair, Lionel Patrone, Mathieu Abel, Louis Porte, Olivier Chuzel and Jean-Luc Parrain Chem. Sci., 2013, 4, 2815-2821

Michael Addition-Initiated Sequential Reactions from 1,3-Dicarbonyls for the Synthesis of Polycyclic Heterocycles

X. Bugaut, D. Bonne, Y. Coquerel, J. Rodriguez, T. Constantieux, Curr. Org. Chem. 2013, 1920-1928.

Directed Studies Towards The Total Synthesis of (+)-13-Deoxytedanolide: Simple and Convenient Synthesis of C8-C16 Fragment

Meiries, S., Bartoli, A., Decostanzi, M., Parrain, J.-L., Commeiras, L., Org. Biomol. Chem., 2013, 11, 4882-4890,

First studies directed towards the diastereoselective synthesis of the BCD tricyclic core of brownin

F. Rodier, F., Parrain, J.-L., Chouraqui, G., Commeiras, L. Org. Biomol. Chem., 2013, 11, 4178-4185,

Enantioselective Organocatalyzed Domino Synthesis of Six-Membered Carbocycles

Sébastien Goudedranche, Wilfried Raimondi, Xavier Bugaut, Thierry Constantieux, Damien Bonne and Jean Rodriguez Synthesis 2013, 1909-1930.

Metal-free Michael addition-initiated three-component reaction for the regioselective synthesis of highly functionalized pyridines: scope, mechanistic investigations and applications

Christophe Allais, Frédéric Liéby-Muller, Thierry Constantieux and Jean Rodriguez Eur. J. Org. Chem. 2013, 2013, 19, 4131-4145.

Tartrate-based ionic liquids: unified synthesis and characterisation

Anne Rouch, Tessa Castellan, Isabelle Fabing, Nathalie Saffon, Jean Rodriguez, Thierry Constantieux, Jean-Christophe Plaquevent and Yves Génisson RSC Adv., 2013, 3, 413-426

Michael Additions in Aqueous Media: 'On-Water' and 'In-Water' Processes from a-Nitroketones and their Anions

G. Giorgi, P. López-Alvarado, S. Miranda, J. Rodriguez, J. C. Menéndez Eur. J. Org. Chem. 2013, 1327.

Diastereoselective Access to Polyoxygenated Polycyclic Spirolactones through a Rhodium-Catalyzed [3+2] Cycloaddition Reaction: Experimental and Theoretical Studies

Fabien Rodier, Michel Rajzmann, Jean-Luc Parrain, Gaëlle Chouraqui, Laurent Commeiras Chem. Eur. J. 2013, 19, 2467-2477.

Cascade Reactions Forming both C-C Bond and C-Heteroatom Bond

D. Bonne, T. Constantieux, Y. Coquerel, J. Rodriguez, dans 'Stereoselective Organocatalysis: Bond Formation Methodologies and Activation Modes', R. Rios Torres, Ed., John Wiley & Sons, Hoboken, New Jersey, 2013, Chap. 16, p. 559-585.

Reactions Involving an alpha,beta-Unsaturated Compound as Electrophilic Component with the Michael Addition as the Key Step

J. Rodriguez, D. Bonne, Y. Coquerel, T. Constantieux, dans 'Multicomponent Reactions 2', 'Science of Synthesis Reference Library', T. J. J. Müller, Ed., Thieme, Stuttgart, 2013, Chap. 2.1.1, p. 1-36.

Microwave-Assisted Stereoselective Synthesis

Y. Coquerel, E. Colacino, J. Rodriguez, J. Martinez, F. Lamaty, in Stereoselective Synthesis of Drugs and Natural Products, Eds: V. Andrushko, N. Andrushko, Wiley- Blackwell, Hoboken, NJ, 2013, Chap. 5, in press. 

Activation of 1,2- and 1,3-Ketoamides with Thiourea Organocatalyst for the Enantioselective Domino Synthesis of Fuctionalized Cyclohexanes

W. Raimondi, M. M. Sanchez Duque, S. Goudedranche, A. Quintard, T. Constantieux, X. Bugaut, D. Bonne, J. Rodriguez Synthesis, 2013, 45, 1659-1666.

Practical and Efficient Organocatalytic Enantioselective ?- Hydroxyamination Reactions of ?-Ketoamides

D. Mailhol, J.-C. Castillo, K. Mohanan, R. Abonia, Y. Coquerel, J. Rodriguez, ChemCatChem 2013, 5, 1192-1199

Stereoselective Multiple Bond-Forming Transformations (MBFTs): The Power of 1,2- and 1,3-Dicarbonyl Compounds

D. Bonne, T. Constantieux, Y. Coquerel, J. Rodriguez, Chem.-Eur. J. 2013, 19, 2218-2231. 

Pt-?catalysed intermolecular hydroamination of non-?activated olefins using a novel family of catalysts: Arbuzov-?type phosphorus metal complexes

Rodrig'uez-Zubiri Mireia, Anguille Stephane, Brunet Jean-Jacques, Daran Jean-Claude, Journal of Molecular Catalysis A: Chemical (2013), 379, 103-111

Syntheses and Applications of Functionalized Bicyclo[3.2.1]octanes: Thirteen Years of Progress

M. Presset, Y. Coquerel, J. Rodriguez, Chem. Rev. 2013, 113, 525-595. 

Organocatalytic Umpolung: N-Heterocyclic Carbenes and Beyond

Xavier Bugaut, Frank Glorius, Chem. Soc. Rev. 2012, 41, 3511-3522.

N-Heterocyclic carbene mediated organocatalytic transfer of tin onto aldehydes: An easy access to syn-diols and mechanistic studies

Romain Blanc, Paola Nava, Michel Rajzman, Laurent Commeiras and Jean-Luc Parrain, Adv. Synth. Catal. 2012, 354, 2038-2048.

Asymmetric Rhodium-Directed anti-Markovnikov Regioselective Boracyclopentannulation

Momar Toure, Olivier Chuzel, and Jean-Luc Parrain J. Am. Chem. Soc. 2012, 134, 17892-17895

Expeditious, Metal-Free, Domino, Regioselective Synthesis of Highly Substituted 2-Carbonyl- and 2-Phosphorylfurans by Formal [3+2] Cycloaddition

Wilfried Raimondi, Daniel Dauzonne, Thierry Constantieux, Damien Bonne, Jean Rodriguez Eur. J. Org. Chem. 2012, 6119-6123.

Expeditious Synthesis of the Cores of Naturally Occurring Cyclic Polyethers using a Divergent Ring Rearrangement Metathesis Strategy

P. Escavabaja, J. Viala, Y. Coquerel, J. Rodriguez, Adv. Synth. Catal., 2012, 354, 3200-3204.

Enantioselective Organocatalytic Michael Addition of Cyclobutanones to Nitroalkenes

D. Mailhol, M. M. Sanchez Duque, W. Raimondi, D. Bonne, T. Constantieux, Y. Coquerel, J. Rodriguez, Adv. Synth. Catal.,2012, 354, 3523-3532.

Dual Heterogeneous Catalysis for a Regioselective Three- Component Synthesis of Bi- and Tri(hetero)arylpyridines

Christophe Allais, Frédéric Liéby-Muller, Thierry Constantieux, Jean Rodriguez Adv. Synth. Catal. 2012, 354 (13), 2537-2544.

Cooperative Heterogeneous Organocatalysis and Homogeneous Metal Catalysis for the One-Pot Regioselective Synthesis of 2-Pyridones

Christophe Allais, Olivier Baslé, Jean-Marie Grassot, Maxime Fontaine, Stéphane Anguille, Jean Rodriguez, Thierry Constantieux Adv. Synth. Catal. 2012, 354 (11-12), 2084-2088.

A Convergent Approach to (-)-Callystatin A Based on Local Symmetry

Mathieu Candy, Loïc Tomas, Sabrina Parat, Virginie Heran, Hugues Bienaymé, Jean-Marc Pons and Cyril Bressy Chem. Eur. J. 2012, 18, 14267-14271

Transition-Metal-Free alpha-Arylation of beta-Keto Amides via an Interrupted Insertion Reaction of Arynes

Kishor Mohanan, Yoann Coquerel, Jean Rodriguez, Org. Lett. 2012, 14, 4686-4689.

Catalyst- and Halogen-Free Regioselective Friedel-Crafts ?-Ketoacylations

Kishor Mohanan, Marc Presset, Damien Mailhol, Yoann Coquerel, Jean Rodriguez Chem. Eur. J. 2012, 18: 9217-9220

Asymmetric transformations involving 1,2-diarbonyl compounds as pronucleophiles

W. Raimondi, D. Bonne, J. Rodriguez, Chem. Commun. 2012, 48, 6763

Dramatic influence of the substitution of alkylidene-5H-furan-2-ones in Diels-Alder cycloadditions with o-quinonedimethide as diene partner: en route to the CDEF polycyclic ring system of lactonamycin

Sébastien Dubois, Fabien Rodier, Romain Blanc, Raphaël Rahmani, Virginie Héran, Jérôme Thibonnet, Laurent Commeiras and Jean-Luc Parrain, Org. Biomol. Chem., 2012, 10, 4712-4719

Microwave-Assisted Domino Benzannulation of ?-Oxo Ketenes: Preparation of 1,3-Dihydro-2H-1,5-benzodiazepin-2-ones

Juan-Carlos Castillo, Marc Presset, Rodrigo Abonia, Yoann Coquerel, Jean Rodriguez Eur. J. Org. Chem. 2012, 2338-2345

Asymmetric organocascades involving the formation of two C-heteroatom bonds from two distinct heteroatoms

Damien Bonne , Thierry Constantieux , Yoann Coquerel andJean Rodriguez, Org. Biomol. Chem., 2012,10, 3969-3973

Activation of 1,2-Ketoesters with Takemoto's Catalyst toward Michael Addition to Nitroalkenes

Wilfried Raimondi, Olivier Baslé, Thierry Constantieux, Damien Bonne, Jean Rodriguez, Adv. Synth. Catal. 2012, 354, 563-568.

Organocatalytic 3+2-Cycloaddition Route to 1,2,3-Triazoles

Victor Snieckus and Benjamin N. Rocke Synfact 2012, 8, 21 (from Mokhtaria Belkheira, Douniazad El Abed, Jean-Marc Pons and Cyril Bressy)

1,2-Dicarbonyl Compounds as Pronucleophiles in Organocatalytic Asymmetric Transformations

Wilfried Raimondi, Damien Bonne, and Jean Rodriguez Angew. Chem. Int. Ed. 2012, 51, 40-42

Collective Domino Approach toward the Core of Molecules Isolated from the Genus Schisandra

Alexandra Bartoli, Gaelle Chouraqui, Jean-Luc Parrain, Org. Lett. 2012, 14, 122-125.

Single-Step Metallocatalyzed and Organocatalyzed Enantioselective Construction of Bicyclo[3.2.1]octanes

M. PRESSET, Y. COQUEREL, J. Rodriguez, ChemCatChem (Highlight) 2012, 4, 172-174.

Access to Polyfunctionalized Diquinanes, Hydrindanes, and Decalines via TiCl4 Promoted Michael-Aldol and Baylis-Hillman Reactions

Ressault, B., Jaunet, A., Geoffroy, P., Goudedranche, S., Miesch, M. Org. Lett., 2012, 14, 366-369.

Stereoselective Multicomponent Reactions: from Simple 1,3-Dicarbonyls to Functionalized Chiral Heterocycles

D. Bonne, Y. Coquerel, T. Constantieux, J. Rodriguez in Targets in Heterocyclic Systems - Chemistry and Properties, Vol. 15, Eds.: O. A. Attanasi, D. Spinelli, Societa? Chimica Italiana, Roma, 2011, pp. 140-163. 

Organo-Click Synthesis of 1,2,3-Triazoles from Unactivated Ketones

Benjamin List and Quinggang Wang Synfact 2011, 12, 1367 (from Mokhtaria Belkheira, Douniazad El Abed, Jean-Marc Pons and Cyril Bressy)

2,6-bis[(4S)-4,5-Dihydro-4-(1-methylethyl)-5,5-diphenyl-2-oxazolyl]pyridine

In electronic Encyclopedia of Organic Reagents (e-EROS), Wiley-VCH, 2011. Auteurs: Arseniyadis, S. and Bressy, C.

N-[(1S)-1-(hydroxydiphenylmethyl)-3-methylbutyl]-2-pyrrolidinecarboxamide

In electronic Encyclopedia of Organic Reagents (e-EROS), Wiley-VCH, 2011. Auteurs: Arseniyadis, S. and Bressy, C.

Organocatalytic Synthesis of 1,2,3-Triazoles from Unactivated Ketones and Arylazides

Mokhtaria Belkheira, Douniazad El Abed, Jean-Marc Pons and Cyril Bressy Chem. Eur. J. 2011, 17, 12917 - 12921

Multicomponent reactions in ionic liquids: convenient and ecocompatible access to the 2,6-DABCO core

Z. El Asri, Y. Génisson, F. Guillen, O. Baslé, N. Isambert, M. M. Sanchez Duque, S. Ladeira, J. Rodriguez, T. Constantieux, J-C. Plaquevent Green Chem., 2011, 13, 2549-2552.

Selected for SYNFACTS by Benjamin List and Manuel Mahlau: Asymmetric Michael Addition of alpha-Substituted beta-Keto Amides

Maria del Mar Sanchez Duque, Olivier Baslé, Nicolas Isambert, Anouk Gaudel-Siri, Yves Génisson, Jean-Christophe Plaquevent, Jean Rodriguez and Thierry Constantieux Synfacts 2011, 8, 0904

1,3-Dipolar Cycloaddition of Hydrazones with ?-Oxo-ketenes: A Three-Component Stereoselective Entry to Pyrazolidinones and an Original Class of Spirooxindoles

Marc Presset, Kishor Mohanan, Marie Hamann, Yoann Coquerel, and Jean Rodriguez Org. Lett. 2011, 13, 4124-4127

Diazo Transfer Reactions to 1,3-Dicarbonyl Compounds with Tosyl azide

Marc Presset, Damien Mailhol, Yoann Coquerel, Jean Rodriguez Synthesis 2011, 2549-2552

A Cooperative Participation of the Amido Group in the Organocatalytic Construction of All-Carbon Quaternary Stereocenters by Michael Addition with beta-Ketoamides

Maria del Mar Sanchez Duque, Olivier Baslé, Nicolas Isambert, Anouk Gaudel-Siri, Yves Génisson, Jean-Christophe Plaquevent, Jean Rodriguez and Thierry Constantieux Org. Lett. 2011, 13, 3296-3299

Consecutive Reactions with Sulfoximines: Straightforward Synthesis of Substituted 5,5-Spiroketals

Vellaisamy Sridharan, Nikolay Vologdin, Marie-Alice Virolleaud, Cyril Bressy, Gaëlle Chouraqui, Laurent Commeiras, Jean-Luc Parrain, Damien Bonne,Yoann Coquerel, Jean Rodriguez Synthesis 2011, 2085-2090.

A General, Diastereoselective Synthesis of Highly Functionalized Bicyclo[n.3.1]alkane Systems Based on an Anionic Domino Reaction of alpha-Nitrocycloalkanones

Giorgio Giorgi, Sonia Miranda, Miriam Ruiz, Jean Rodriguez, Pilar López-Alvarado, and J. Carlos Menéndez Eur. J. Org. Chem. 2011, 2101-2110.

Carboxylate-Directed Tandem Functionalisations of ?,?-Dihaloalkenoic Acids with 1-Alkynes: A Straightforward Access to (Z)-Configured, ?,?-Substituted ?-Alkylidenebutenolides

Samuel Inack?Ngi, Khalil Cherry, Virginie Héran, Laurent Commeiras, Jean-Luc Parrain, Alain Duchêne, Mohamed Abarbri, Jérôme Thibonnet Chemistry - A European Journal 2011, 17 (49), 13692-13696

Construction of spirolactones with concomitant formation of the fused quaternary centre - application to the synthesis of natural products

Alexandra Bartoli, Fabien Rodier, Laurent Commeiras, Jean-Luc Parrain and Gaelle Chouraqui, Nat. Prod. Rep. 2011, 28, 763-782.

Multicomponent reactions and ionic liquids: a perfect synergy for eco-compatible heterocyclic synthesis

N. Isambert, M. M. Sanchez Duque, J.-C. PLaquevent, Y. Génisson, J. Rodriguez, T. Constantieux, Chem. Soc. Rev., 2011, 40, 1347-1357.

N-Heterocyclic Carbene-Catalyzed Michael Additions of 1,3-Dicarbonyl Compounds

T. Boddaert, Y. Coquerel, J. Rodriguez, Chem. Eur. J. 2011, 17, 2266-2271.

Expeditious Divergent Synthetic Approach to Polycyclic Terpene-like Molecules

T. Boddaert, Y. Coquerel, J. Rodriguez, Chem. Eur. J. 2011, 17, 2048-2051.

Exploiting the Divergent Reactivity of a-Isocyanoacetate: Multicomponent Synthesis of 5-Alkoxyoxazoles and Related Heterocycles

Claudia Lalli, Marinus J. Bouma, Damien Bonne, Géraldine Masson, and Jieping Zhu Chem. Eur. J. 2011, 17, 880 - 889.

The Shortest Synthetic Route to Puromycin Analogues Using a Modified Robins Approach

Krishnakumar, K. S., Goudedranche, S., Bouchu D., Strazewski, P. J. Org. Chem., 2011, 76, 2253-2256.

Relative Stability of a Series of 1,2,3-Triazolines. Theoretical Study of Substituent Effects

Hamadouche, M., Gaudel-Siri, A., Pons, J.-M., El Abed, D J. Mol. Struct. (Theochem) 2010, 33-37.

Expeditious Synthesis and Biological Evaluation of New C-6 1,2,3-Triazole Adenosine Derivatives A1 Receptor Antagonists or Agonists

Smitha C. Mathew, Youlet By, Aurélie Berthault, Marie-Alice Virolleaud, Louis Carrega, Gaëlle Chouraqui, Laurent Commeiras, Jocelyne Condo, Mireille Attolini, Anouk Gaudel-Siri, Jean Ruf, Jean Rodriguez, Jean-Luc Parrain and Régis Guieu Org. Biomol. Chem. 2010, 8, 3874-3881

Highly diastereo- and enantioselective organocatalytic Micheal addition of a-ketoamides to nitroalkenes

O. Baslé, W. Raimondi, M. M. Sanchez Duque, D. Bonne, T. Constantieux, J. Rodriguez. Org. Lett., 2010, 12, 5246-5249.

Diels-Alder cycloaddition of o-quinonedimethides and alkylidene-5H-furan-2-ones: New and rapid access to lambertellol cores and arthrinone derivatives.

Blanc, R., Heran, V., Rahmani, R., Commeiras, L., Parrain, J.-L. Org. Biomol. Chem. 2010, 8, 5490-5494.

One-pot asymmetric cyclocarbohydroxylation sequence for the enantioselective synthesis of functionalised cyclopentanes

Wilfried Raimondi, Grégory Lettieri, Jean-Pierre Dulcère, Damien Bonne and Jean Rodriguez Chem, Commun, 2010, 46, 7247-7249.

A syntheis of (-)-ebelactones A and B

J.P. Cooksey, R Ford, P.J. Kocienski, B. Pelotier, J.-M. Pons Tetrahedron 2010, 66, 6462-6467.

alpha- and beta-Stannyl Trifluoromethylbutenoates: Regioselective Preparation and Use in Copper(I)-Catalyzed Allylation and Propargylation Reactions

Yvan Carcenac, Khalid Zine, Jean-Claude Kizirian, Jérôme Thibonnet, Alain Duchêne, Jean-Luc Parrain, Mohamed Abarbri Advanced Synthesis & Catalysis Volume 352, Issue 6, Date: April 19, 2010, Pages: 949-954

Domino allylic amination/Sonogashira/heterocyclisation reactions: palladium-catalysed three-component synthesis of pyrroles

Sandrine Lamandé-Langle, Mohamed Abarbri, Jérôme Thibonnet, Alain Duchêne and Jean-Luc Parrain, Chem. Commun. 46, 5157-5159.

Utilisation des dérivés 1,3-dicarbonylés dans les réactions domino et multicomposé

Damien Bonne, Thierry Constantieux, Yoann Coquerel, Jean Rodriguez Techniques de l'Ingénieur 2010, CHV2210

1,3-Dicarbonyl compounds in stereoselective domino and multicomponent reactions

Damien Bonne, Yoann Coquerel, Thierry Constantieux, Jean Rodriguez Tetrahedron: Asymmetry 2010, 21, 1085-1109

beta-diketo building blocks for MCRs-based syntheses of heterocycles

M.M. Sanchez Duque, C. Allais, N. Isambert, T. Constantieux, J. Rodriguez Top. Heterocyclic. Chem. 2010, 23, 227-277

Quadrane Sesquiterpenes: Natural Sources, Biology, and Syntheses

Marc Presset, Yoann Coquerel, Jean Rodriguez Eur. J. Org. Chem. (microreview) 2010, 2247-2260.

Total Synthesis of (+)-Crocacin C Using Hidden Symmetry

Mathieu Candy, Gérard Audran, Hugues Bienaymé, Cyril Bressy, and Jean-Marc Pons J. Org. Chem. 2010, 75, 1354-1359 (featured article and highlighted by Synfacts 2010, 7, 744).

Multiple Bond-Forming Transformations: the Key Concept towards Eco-compatible Synthetic Organic Chemistry

Yoann Coquerel, Thomas Boddaert, Marc Presset, Damien Mailhol, Jean Rodriguez in Ideas in Chemistry and Molecular Sciences, Vol.1 Advances in synthetic chemistry, Chap 9, pp 187-202, Pignataro B. Ed., Wiley-VCH, Weinheim, 2010.

Design, synthesis and biological evaluation of bivalent m opiate and adenosine A1 receptor antagonist.

S. C. Mathew, N. Ghosh, Y. By, A. Berthault, M. A. Virolleaud, L. Carrega, G. Chouraqui, L. Commeiras, J. Condo, M. Attolini, A. gaudel-SIRI, J. Ruf, J. L. Parrain, J. Rodriguez, R. Guieu, Bioorg. Med. Chem. Lett. 2009, 19, 6736-6739.

Michael Addition Initiated Carbocyclization Sequences with Nitroolefins for the Stereoselective Synthesis of Functionalized Heterocyclic and Carbocyclic Systems

Estelle Dumez, Anne-Catherine Durand, Martial Guillaume, Pierre-Yves Roger, Robert Faure, Jean-Marc Pons, Gaetan Herbette, Jean-Pierre Dulcere, Damien Bonne, and Jean Rodriguez Chem. Eur. J. 2009, 15, 12470-2488

Use of beta,gamma-Unsaturated alpha-Ketocarbonyls for a Totally Regioselective Oxidative Multicomponent Synthesis of Polyfunctionalized Pyridines

Christophe Allais, Thierry Constantieux and Jean Rodriguez, Chem. Eur. J. 2009, 15, 12945-12948.

Enantioselective Enzymatic Desymmetrization of Highly Functionalized Meso Tetrahydropyranyl Diols

Mathieu Candy, Gérard Audran, Hugues Bienaymé, Cyril Bressy, and Jean-Marc Pons Org. Lett. 2009, 4950-4953

Consecutive reactions with sulfoximines: A direct access to 2-sulfonimidoylylidene tetrahydrofurans and 6-sulfonimidoylmethyl-3,4-dihydro-2H-pyrans

M.-A. Virolleaud, V. Sridharan, D. Mailhol, D. Bonne, C. Bressy, G. Chouraqui, L. Commeiras, Y. Coquerel, J. Rodriguez Tetrahedron, 2009, 65, 9756-9764.

Highly efficient synthesis of trans-beta,gama-unsaturated-alpha-keto amides

Christophe Allais, Thierry Constantieux, and Jean Rodriguez synthesis 2009, 2523-2530,

User friendly stereoselective one-pot access to 1,4-diazepane derivatives by a cyclodehydrative three-component reaction with 1,3-dicarbonyls

Enrique Sotoca, Christophe Allais, Thierry Constantieux, Jean Rodriguez Org. Biomol. Chem., 2009, 7, 1911-1920

Studies Towards the Total Synthesis of (-)-Caulerpenynol, a Toxic Sesquiterpenoid of the Green Seaweed Caulerpa taxifolia

Laurent Commeiras, L., Thibonnet, J., Parrain, J.-L. Eur. J. Org. Chem., 2009, 2987-2997

Caulerpenyne Binding to Tubulin: Structural Modifications by a Non Conventional Pharmacological Agent

Bourdron, J., Barbier, P., Allegro, D., Villard, C., Lafitte, D., Commeiras, L., Parrain, J.-L., Peyrot, V. Medecinal chemistry, 2009, 5, 182-190

Copper-Catalyzed Preparation of -Alkylidenebutenolides and Isocoumarins under Mild Palladium-Free Conditions

Inack-Ngi S., Rahmani R., Commeiras L., Chouraqui G., Thibonnet J., Duchêne A., Abarbri M., Parrain J.-L. Adv. Synth. Catal. 2009, 351, 779 - 788

Microwave-assisted Cross-metathesis of Acrylonitrile

Thomas Boddaert, Yoann Coquerel, Jean Rodriguez C. R. Chimie 2009, 12, 872-875.

First Total Synthesis of (-)-Caulerpenynol

Commeiras, L., Thibonnet, J., Parrain, J.L. Org. Biomol. Chem., 2009,7, 425-427.

Palladium-Catalysed Isomerisation of 2-Vinylidenehydrofurans into 1,3-Dienes and some Aspects of their Reactivity

Abdelkader Ghobsi, Salih Hacini, Laurence Wavrin, Anouk Gaudel-Siri, Agnès Corbères, Cyril Nicolas, Damien Bonne, Jacques Viala, and Jean Rodriguez Eur. J. Org. Chem. 2008, 4446-4453

Microwave-Assisted Olefin Metathesis

Yoann Coquerel, Jean Rodriguez Eur. J. Org. Chem. (microreview) 2008, 1125-1132

Aldolisation and carboxylation reactions from ?-silyl-?-lactams. A combined theoretical and experimental study

Sabrina Parat, S., Pelotier, B., Fournier, L., Rajzmann, M., Kocienski, P.J. , Pons, J.-M. Heterocycle 2008, 70, 2429-2441

Synthetic Studies Towards Guaianolide Sesquiterpene Lactones

Isabelle Reboul, Thomas Boddaert, Yoann Coquerel, Jean Rodriguez Eur. J. Org. Chem. 2008, 5379-5382

Stereoselective Synthesis of Bicyclo[4.2.1]nonanes: a Temporary-Bridge Approach to Cyclooctanoids

Antoine Michaut, Sonia Miranda-García, J. Carlos Menéndez,Yoann Coquerel, Jean Rodriguez Eur. J. Org. Chem. 2008, 4988-4998.

Metal-free Michael addition initiated multicomponent oxidative cyclodehydration route to polysubstituted pyridines from 1,3-dicarbonyls

Frédéric Liéby-Muller, Christophe Allais, Thierry Constantieux and Jean Rodriguez, Chem. Commun., 2008, 4207-4209

Catalytic Properties of the Pd/C - Triethylamine System

Yoann Coquerel, Jean Rodriguez Arkivoc 2008 (xi) 227-237.

Bicyclic 5-6 Systems with One Bridgehead (Ring Junction) Nitrogen Atom: Two Extra Heteroatoms 0:2

J. Rodriguez, T. Constantieux. Comprehensive Heterocyclic Chemistry III, AR Katritzky, CA Ramsden, EFV Scriven and RJK Taylor, Eds., Elsevier: Oxford, 2008, Vol. 11, pp 629 - 644.

The MARDi cascade : A Michael-Initiated Domino-Multicomponent Approach for the Stereoselective Synthesis of Seven-Membered Rings

Y. Coquerel, M.-H. Filippini, D. Bensa, J. Rodriguez Chem. Eur. J. 2008, 14, 3078-3092

Straightforward one-pot stereoselective synthesis of substituted tetrahydrofurans from 1,3-butadienes and aldehydes.

M. Roux, C. Aouf, J. -L. Parrain et M. Santelli, Tetrahedron Lett. 2007, 48, 4011-4014.

First Total Synthesis and Assignment of the Stereochemistry of Crispatenine

Julien Bourdron, Laurent Commeiras,Gérard Audran, Nicolas Vanthuyne, J. C. Hubaud, Jean-Luc Parrain J. Org. Chem 2007, 72, 3770-3775.

Selective Synthesis of b-hydroxy Nitroethanol Ethers by Alcoholysis of Oxiranes

Gras, J.-L, Daoubi, M., Collado, I. Synthetic Comm. 2007, 37:20, 3589 - 3598

Reluctant Cross-Metathesis Reactions: a Highly Beneficial Effect of Microwave Irradiation

Michaut, A,, Boddaert, T., Coquerel, Y., Rodriguez, J. Synthesis 2007, 2867-2871

Pd-H from Pd/C and Triethylamine: Implications in Palladium Catalysed Reactions Involving Amines

Coquerel, Y., Brémond, P., Rodriguez, J. J. Organomet. Chem. 2007, 692, 4805-4808.

Stereoselective Synthesis of the Core of Naturally Occurring Anti-HIV Isolitseane B

Brémond, P., Girardeau, E., Coquerel, Y., Rodriguez Lett. Org. Chem. 2007, 4, 232-233